Patent application number | Description | Published |
20080319020 | 4-Oxadiazolyl-Piperidine Compounds and Use Thereof -
4-Oxadiazolyl-piperidine compounds of formula (I) and (II), their compositions and use for the treatment of pain and diarrhoea. | 12-25-2008 |
20090105249 | 4-phenylsulfonamidopiperidines as calcium channel blockers -
The invention relates to piperidinyl compounds of Formula (I): or a pharmaceutically acceptable salt, prodrug, or solvate thereof, wherein R | 04-23-2009 |
20090118319 | Fused and Spirocycle Compounds and the Use Thereof - The invention relates to fused and spirocycle compounds of Formula (I), or a pharmaceutically acceptable salt, prodrug, or solvate thereof, wherein R | 05-07-2009 |
20090170868 | TRPV1 ANTAGONISTS INCLUDING DIHYDROXY SUBSTITUENT AND USES THEREOF - The invention relates to compounds of formula IA | 07-02-2009 |
20090176796 | TRPV1 ANTAGONISTS INCLUDING AMIDE SUBSTITUENT AND USES THEREOF - The invention relates to compounds of formula IA″ | 07-09-2009 |
20100004254 | THERAPEUTIC AGENTS USEFUL FOR TREATING PAIN - A compound of formula: | 01-07-2010 |
20100120862 | MONOCYCLIC COMPOUNDS AND THEIR USE AS TRPV1 LIGANDS - The invention relates to compounds of formula I | 05-13-2010 |
20100130499 | BICYCLOHETEROARYL COMPOUNDS AND THEIR USE AS TRPV1 LIGANDS - The invention relates to compounds of formula I | 05-27-2010 |
20100130552 | Therapeutic Agents Useful for Treating Pain - A compound of Formula: (I) or a pharmaceutically acceptable derivative thereof, where Ar | 05-27-2010 |
20100137306 | HETEROCYCLIC TRPV1 RECEPTOR LIGANDS - The invention relates to compounds of formulae I(a)-I(d): | 06-03-2010 |
20110136833 | Tetrahydropyridinyl and Dihydropyrrolyl Compounds and the Use Thereof - The invention relates to tetrahydropyridinyl and dihydropyrrolyl compounds of Formula (I): and pharmaceutically acceptable salts, prodrugs, or solvates thereof, wherein X, Y, Z, R | 06-09-2011 |
20110281885 | THERAPEUTIC AGENTS USEFUL FOR TREATING PAIN - A compound of formula: | 11-17-2011 |
20120004217 | THERAPEUTIC AGENTS USEFUL FOR TREATING PAIN - A compound of formula: | 01-05-2012 |
20120015954 | THERAPEUTIC AGENTS USEFUL FOR TREATING PAIN - A compound of formula: | 01-19-2012 |
20120177570 | TRPV1 ANTAGONISTS INCLUDING AMIDE SUBSTITUENT AND USES THEREOF - The invention relates to compounds of formula IA″ | 07-12-2012 |
20120309778 | Fused and Spirocycle Compounds and the Use Thereof - The invention relates to fused and spirocycle compounds of Formula (I), or a pharmaceutically acceptable salt, prodrug, or solvate thereof, wherein R | 12-06-2012 |
20130150377 | Tetrahydropyridinyl and Dihydropyrrolyl Compounds and the Use Thereof - The invention relates to tetrahydropyridinyl and dihydropyrrolyl compounds of Formula (I): and pharmaceutically acceptable salts, prodrugs, or solvates thereof, wherein X, Y, Z, R | 06-13-2013 |
20130289044 | Quinazoline Compounds as Sodium Channel Blockers - The invention relates to aryl substituted quinazolines of Formula I, and pharmaceutically acceptable salts, prodrugs, or solvates thereof, wherein G, A, and R | 10-31-2013 |
20130296281 | Aryl Substituted Indoles and Their Use as Blockers of Sodium Channels - The invention relates to aryl and heteroaryl substituted compounds of Formula (I), and pharmaceutically acceptable salts, prodrugs, or solvates thereof, wherein G, R | 11-07-2013 |
20130303526 | Pyridine Compounds and the Uses Thereof - The invention relates to substituted pyridine compounds of Formula (I) and the pharmaceutically acceptable salts, prodrugs, and solvates thereof, wherein R | 11-14-2013 |
20130338170 | TRPV1 ANTAGONISTS INCLUDING DIHYDROXY SUBSTITUENT AND USES THEREOF - The invention relates to compounds of formula IA | 12-19-2013 |
20130345211 | Pyridine Compounds as Sodium Channel Blockers - The invention relates to substituted pyridine compounds of Formula I: (I) or a pharmaceutically acceptable salt, prodrug, or solvate thereof wherein A | 12-26-2013 |
20140005212 | Substituted Pyridines as Sodium Channel Blockers | 01-02-2014 |
20140045875 | Fused and Spirocycle Compounds and the Use Thereof - The invention relates to fused and spirocycle compounds of Formula (I), or a pharmaceutically acceptable salt, prodrug, or solvate thereof, wherein R | 02-13-2014 |
20140057931 | BUPRENORPHINE ANALOGS - The present invention is directed to Buprenorphine Analog compounds of the Formula (I), Formula (IA) or Formula (IB) shown below, wherein R | 02-27-2014 |
20140128346 | PHOSPHORUS-SUBSTITUTED QUINOXALINE-TYPE PIPERIDINE COMPOUNDS AND USES THEREOF - The disclosure relates to Phosphorus-Substituted Quinoxaline-Type Piperidine Compounds of Formula (I): | 05-08-2014 |
20140135351 | Benzomorphan Analogs and the Use Thereof - The present invention is directed to Benzomorphan Analog compounds of the Formula I″, Formula IA″, Formula IB″, Formula IC″, or Formula ID″ as shown below; and related Formula I′, Formula IA′, Formula IB′, Formula IC′, or Formula ID′; Formula I, Formula IA, Formula IB, Formula IC, or Formula ID; wherein R | 05-15-2014 |
20140142112 | THERAPEUTIC AGENTS USEFUL FOR TREATING PAIN - A compound of formula: | 05-22-2014 |
20140171461 | Nitrogen Containing Morphinan Derivatives and the Use Thereof - The application is directed to compounds of Formula I-A | 06-19-2014 |
20140179724 | Spirocyclic Morphinans and Their Use - The application is directed to compounds of Formula I′-A | 06-26-2014 |
20140187571 | 7,8-Cyclicmorphinan Analogs - The application is directed to compounds of Formula I-A | 07-03-2014 |
20140187573 | Substituted Morphinans and the Use Thereof - The application is directed to compounds of Formula I: | 07-03-2014 |
20140221419 | BENZOMORPHAN ANALOGS AND THE USE THEREOF - The present invention is directed to Benzomorphan Analog compounds of the Formula I-ID as shown below, wherein R | 08-07-2014 |
20140249159 | HETEROCYCLIC COMPOUNDS - The invention relates to compounds of Formula I: wherein Ar | 09-04-2014 |
20140275117 | BUPRENORPHINE ANALOGS - The present invention is directed to Buprenorphine Analog compounds of Formula I, II, III, IV or V and including various stereoisomers (such as Formula IA shown below), wherein R | 09-18-2014 |
20140303139 | PYRIMIDINES AS SODIUM CHANNEL BLOCKERS - The present disclosure provides substituted pyrimidine compounds of Formula (I), and the pharmaceutically acceptable salts, prodrugs, and solvates thereof, wherein A | 10-09-2014 |
20140329829 | TRPV1 ANTAGONISTS INCLUDING DIHYDROXY SUBSTITUENT AND USES THEREOF - The disclosure relates to Compounds of Formula (I) | 11-06-2014 |
20150018366 | TRPV1 ANTAGONISTS INCLUDING DIHYDROXY SUBSTITUENT AND USES THEREOF - The invention relates to compounds of formula IA | 01-15-2015 |
20150045397 | SUBSTITUTED PYRIDINES AS SODIUM CHANNEL BLOCKERS - The invention relates to substituted pyridine and pyrimidine compounds of Formula (I) and the pharmaceutically acceptable salts, prodrugs, and solvates thereof, wherein R | 02-12-2015 |
20150057300 | SUBSTITUTED PIPERIDINES AS SODIUM CHANNEL BLOCKERS - The present disclosure provides substituted piperidines or pyrrolidines having Formula IA: | 02-26-2015 |