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Kurt Gordon Pike, Cheshire GB

Kurt Gordon Pike, Cheshire GB

Patent application numberDescriptionPublished
20080234273Heteroaryl Benzamide Derivatives for Use as Glk Activators in the Treatment of Diabetes - Compounds of formula (I)09-25-2008
20080280872Benzamide Derivatives and Their Use as Glucokinase Activating Agents - Compounds of Formula (I): wherein: R11-13-2008
20080280874Phenoxy Benzamide Compounds with Utility in the Treatment of Type 2 Diabetes and Obesity - Compounds of Formula (I):11-13-2008
20080312207Compounds - Compounds of Formula (I) wherein: R1 is methyl; R2 is selected from —C (O) NR4R5, SO2NR4R5, S (O) pR4 and HET-2; HET-1 is a 5- or 6-membered, optionally substituted C-linked heteroaryl ring; HET-2 is a 4-, 5- or 6-membered, C- or N-linked optionally substituted heterocyclyl ring; R3 is selected from halo, fluoromethyl, difluoromethyl, trifluoromethyl, methyl, methoxy and cyano; R4 is selected from for example hydrogen, optionally substituted (1-4C) alkyl and HET-2; R5 is hydrogen or (1-4C) alkyl; or R4 and R5 together with the nitrogen atom to which they are attached may form a heterocyclyl ring system as defined by HET-3; HET-3 is for example an optionally substituted N-linked, 4, 5 or 6 membered, saturated or partially unsaturated heterocyclyl ring; p is (independently at each occurrence) 0, 1 or 2; m is 0 or 1; n is 0, 1 or 2; provided that when m is 0, then n is 1 or 2; or a salt, pro drug or solvate thereof, are described. Their use as GLK activators, pharmaceutical compositions containing them and processes for their preparation are also described.12-18-2008
20090018157Chemical compounds - Compounds of Formula (I) wherein: R01-15-2009
20090029905HETEROARYL BENZAMIDE DERIVATIVES FOR USE AS GLK ACTIVATORS IN THE TREATMENT OF DIABETES - Compounds of formula (I)01-29-2009
20090062351Benzoyl amino pyridyl carboxylic acid derivatives useful as glucokinase (glk) activators - A compound of Formula (I): Formula (I) wherein: R03-05-2009
20090105214Heteroaryl Benzamide Derivatives for Use as Glk Activators in the Treatment of Diabetes - Compounds of formula (I), wherein R04-23-2009
20090105263HETEROBICYCLIC COMPOUNDS AS GLUCOKINASE ACTIVATORS - Compounds of Formula (I):04-23-2009
20090118159HETEROARYL BENZAMIDE DERIVATIVES FOR USE AS GLK ACTIVATORS IN THE TREATMENT OF DIABETES - Compounds of formula (I)05-07-2009
20090253676Heteroaryl Benzamide Derivatives for Use as GLK Activators in the Treatment of Diabetes - Compounds of Formula (I):10-08-2009
20090264336HETEROARYL BENZAMIDE DERIVATIVES FOR USE AS GLK ACTIVATORS IN THE TREATMENT OF DIABETES - Compounds of formula (I)10-22-2009
201100539102 -HETEROCYCLYLOXYBENZOYL AMINO HETEROCYCLYL COMPOUNDS AS MODULATORS OF GLUCOKINASE FOR THE TREATMENT OF TYPE 2 DIABETES - Compounds of formula (I)03-03-2011
201100599412-PHENYL SUBSTITUTED IMIDAZOL [4,5B] PYRIDINE/PYRAZINE AND PURINE DERIVATIVES AS GLUCOKINASE MODULATORS - Compounds of Formula (I), wherein R03-10-2011

Patent applications by Kurt Gordon Pike, Cheshire GB