| Patent application number | Description | Published |
|---|
| 20080207900 | TWO CYCLIC OXOMORPHORIN DERIVATIVES - The present invention relates to a compound represented by formula (I): | 08-28-2008 |
| 20080227815 | Crystal of Indole Derivative Having Piperidine Ring and Process for Production Thereof - A crystal of 1-[1-[2-(7-methoxy-2,2-dimethyl-4-oxochroman-8-yl)-ethyl]piperidin-4-yl]-N-methyl-1H-indole-6-carboxamide fumarate which has peaks at chemical shifts of about 124.0 ppm and about 26.8 ppm in a | 09-18-2008 |
| 20090048213 | Prodrug of cinnamide compound - The present invention provides a most suitable prodrug of a cinnamide compound. The prodrug is represented by Formula (I) | 02-19-2009 |
| 20090048448 | SALTS OF CYNNAMIDE COMPOUND OR SOLVATES THEREOF - The invention provides crystals of dihydrochloride monohydrate of the compound of the following formula having an Aβ production inhibiting effect which crystals are characterized by exhibiting a diffraction peak at an angle of diffraction (2θ±0.2°) of 10.9° in powder X-ray diffractometry. Further, the invention also provides the compound in the form of various salts, crystal forms and amorphous forms which are suitable for the development of drugs. | 02-19-2009 |
| 20090062529 | MULTI-CYCLIC COMPOUNDS - A compound represented by the formula (I): | 03-05-2009 |
| 20090181945 | TWO CYCLIC CINNAMIDE COMPOUND - The present invention relates to a novel two cyclic cinnamide compound and a pharmaceutical agent comprising the compound as an active ingredient. The two cyclic cinnamide compound represented by the general formula (I): | 07-16-2009 |
| 20090203697 | HETEROCYCLIC TYPE CINNAMIDE DERIVATIVE - Disclosed is a compound represented by the formula (I) below or a pharmacologically acceptable salt thereof. Also disclosed is a use of the compound or salt as a pharmaceutical product. | 08-13-2009 |
| 20090203916 | Amorphous object of cinnamide compound - An amorphous object of (3E)-1-[l(s)-1-(4-fluorophenyl)ethyl]-3-[3-methoxy-4-(4methyl-1H-imidazol-1-yl)benzylidene]piperidine-2-one, which is represented by the formula (1) and has Aβ-production inhibitory activity. The amorphous object has such satisfactory properties that it has excellent solubility, is stable, does not readily become a crystalline form, and has low hygroscopicity. It is hence suitable for use in pharmaceutical preparations. | 08-13-2009 |
| 20090281310 | CINNAMIDE COMPOUND - The present invention relates to a process for preparing a compound of formula (6a): | 11-12-2009 |
| 20100105904 | UREA TYPE CINNAMIDE DERIVATIVE - Disclosed is a compound represented by the formula (I) below or a pharmacologically acceptable salt thereof. Also disclosed is a use of the compound or salt as a pharmaceutical product. | 04-29-2010 |
| 20100113773 | BICYCLIC OXOMORPHOLINE DERIVATIVE - The present invention relates to a compound represented by formula (I): | 05-06-2010 |
| 20100168095 | MULTI-CYCLIC CINNAMIDE DERIVATIVES - The present invention provides a compound represented by the formula (I): | 07-01-2010 |
| 20100197926 | METHOD FOR PRODUCING INDOLE DERIVATIVE HAVING PIPERIDINE RING - It is possible to commercially advantageously prepare 1-{1-[2-(7-methoxy-2,2-dimethyl-4-oxochroman-8-y)ethyl]piperidin-4-yl}-N-methyl-1H-indole-6-carboxamide by coupling (7-methoxy-2,2-dimethyl-4-oxochroman-8-yl)acetaldehyde, which is obtained by oxidizing 8-(2-hydroxyethyl)-7-methoxy-2,2-dimethylchroman-4-one, with N-methyl-1-(piperidin-4-yl)-1H-indole-6-carboxamide. | 08-05-2010 |
| 20100324297 | METHOD FOR PRODUCING 1, 2-DIHYDROPYRIDINE-2-ONE COMPOUND - The present inventions provide a method for commercially producing a 1,2-dihydropyridine-2-one compound represented by the following formula (III-a) | 12-23-2010 |
| 20110009619 | POLYCYCLIC COMPOUND - Disclosed is a compound represented by the formula (I): | 01-13-2011 |
| 20110065696 | IMIDAZOYL PYRIDINE COMPOUNDS AND SALTS THEREOF - A compound represented by the formula (I): | 03-17-2011 |
| 20110086860 | COMPOUND - A compound represented by Formula (I) is provided: | 04-14-2011 |
| 20110112138 | MULTI-CYCLIC CINNAMIDE DERIVATIVES - The present invention provides a compound represented by the formula (I): | 05-12-2011 |
