Patent application number | Description | Published |
20080261957 | DIHYDRO-BENZO[B][1,4]DIAZEPIN-2-ONE SULFONAMIDE DERIVATIVES - The present invention relates to compounds of formula (I), a process for the manufacture thereof, their use for the preparation of medicaments for treating CNS disorders and pharmaceutical compositions containing them. Compounds of formula (I) are represented by general formula (I) | 10-23-2008 |
20080280924 | PYRIDINE AND PYRIMIDINE DERIVATIVES AS MGLUR2 ANTAGONISTS - The present invention relates to compounds of formula (I) | 11-13-2008 |
20080300250 | ACETYLENYL-PYRAZOLO-PYRIMIDINE DERIVATIVES - The present invention relates to compounds of formula (I): | 12-04-2008 |
20090088451 | QUINOLINES - The present invention relates to 2-aminoquinolines of formula I | 04-02-2009 |
20090143580 | SUBSTITUTED PYRAZOLO [1,5-a] PYRIMIDINES AS METABOTROPIC GLUTAMATE ANTAGONISTS - The present invention relates to compounds of formula (I) | 06-04-2009 |
20090318474 | PYRIDINE AND PYRIMIDINE DERIVATIVES AS MGLUR 2 ANTAGONISTS - The present invention relates to compounds of formula (I), a process for the manufacture thereof, pharmaceutical compositions containing them, and their use for treating CNS disorders: | 12-24-2009 |
20100063037 | 6-SUBSTITUTED BENZOXAZINES - The present invention is concerned with 6-substituted benzoxazine derivatives of formula (I) | 03-11-2010 |
20100063042 | 5-SUBSTITUTED BENZOXAZINES - The present invention is concerned with 5-substituted benzoxazine derivatives of formula (I) | 03-11-2010 |
20100210642 | ACETYLENYL-PYRAZOLO-PYRIMIDINE DERIVATIVES - The present invention relates to compounds of formula (I): | 08-19-2010 |
20100227887 | PYRIDINE-2-YL CARBOXYLIC ACID AMIDES - The present invention relates to pyridine-2-yl-carboxylic acid amides which act as metabotropic glutamate receptor antagonists. In particular, the present invention relates to pyridine-2-yl-carboxylic acid amides of formula I | 09-09-2010 |
20110015202 | IMIDAZOLES - The present invention relates to imidazole derivatives of the general formula | 01-20-2011 |
20110263615 | PYRIDINE AND PYRIMIDINE DERIVATIVES AS MGLUR2 ANTAGONISTS - The present invention relates to compounds of formula (I) | 10-27-2011 |
20110313151 | ANELLATED PYRIDINE COMPOUNDS - The present invention is concerned with novel dual modulators of the 5-HT | 12-22-2011 |
20120010201 | NOVEL ANELLATED PYRIDINE COMPOUNDS - The present invention is concerned with novel dual modulators of the 5-HT | 01-12-2012 |
20120041002 | SUBSTITUTED PYRAZOLO [1,5-A] PYRIMIDINES AS METABOTROPIC GLUTAMATE ANTAGONISTS - The present invention relates to compounds of formula (I) | 02-16-2012 |
20120136018 | QUINOLINES - The present invention relates to 2-aminoquinolines of formula I | 05-31-2012 |
20120157449 | BENZOFURANE COMPOUNDS - The present invention is concerned with novel dual modulators of the 5-HT | 06-21-2012 |
20120225868 | NOVEL BENZODIOXOLE PIPERIDINE COMPOUNDS - The present invention is concerned with novel dual modulators of the 5-HT | 09-06-2012 |
20120283254 | NOVEL BENZOFURANE-PIPERIDINE COMPOUNDS - The present invention is concerned with novel selective dual modulators of the 5-HT | 11-08-2012 |
20130040948 | NOVEL BENZODIOXOLE PIPERAZINE COMPOUNDS - The present invention is concerned with novel dual modulators of the 5-HT | 02-14-2013 |
20130085278 | METHODS FOR THE PREPARATION OF 5-[2-[7 (TRIFLUOROMETHYL)-5-[4- (TRIFLUOROMETHYL)PHENYL]PYRAZOLO [1,5-A]PYRIMIDIN-3-YL]ETHYNYL]-2-PYRIDINAMINE - The present invention provides methods for preparing 5-[2-[7-(trifluoromethyl)-5-[4-(trifluoromethyl)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]ethynyl]-2-pyridinamine (compound A), which is useful for the treatment of depression and other CNS disorders. The present methods are useful for preparing compound A on large scale in manufacturing facilities. | 04-04-2013 |