Patent application number | Description | Published |
20080234334 | 1,4 DIAMINO BICYCLIC RETIGABINE ANALOGUES AS POTASSIUM CHANNEL MODULATORS - This invention is directed to compounds of formula I, | 09-25-2008 |
20080306063 | PHENYLAMINO ISOTHIAZOLE CARBOXAMIDINES AS MEK INHIBITORS - The invention concerns compounds which inhibit MEK and which have activity as anti-neoplastic agents. These compounds include N-substituted-3-hydroxy-5-arylamino-isothiazole-4-carboxamidines. Also included are the tautomeric isothiazol-3(2H)-ones. | 12-11-2008 |
20090029983 | NOVEL HETEROCYCLIC COMPOUNDS HAVING ANTI-HBV ACTIVITY - This application relates to novel fused tricyclic thienopyridines of Formulas I and II, which useful for treating Hepatitis B infection and other diseases. | 01-29-2009 |
20090137041 | 3-HYDROXYISOTHIAZOLE-4-CARBOXAMIDINE DERIVATIVES AS CHK2 INHIBITORS - This invention provides compounds of Formula I | 05-28-2009 |
20090137635 | DERIVATIVES OF 5-AMINO-4,6-DISUBSTITUTED INDOLE AND 5-AMINO-4,6-DISUBSTITUTED INDOLINE AS POTASSIUM CHANNEL MODULATORS - This invention provides compounds of formula I | 05-28-2009 |
20090326059 | BENZYLOXY ANILIDE DERIVATIVES USEFUL AS POTASSIUM CHANNEL MODULATORS - The present invention relates to benzyloxyanilide derivatives having the following structural formula: | 12-31-2009 |
20110003850 | DERIVATIVES OF 4-(N-AZACYCLOALKYL) ANILIDES AS POTASSIUM CHANNEL MODULATORS - This invention provides a compound of formula IA | 01-06-2011 |
20110118318 | DERIVATIVES OF 5-AMINO-4,6-DISUBSTITUTED INDOLE AND 5-AMINO-4,6-DISUBSTITUTED INDOLINE AS POTASSIUM CHANNEL MODULATORS - This invention provides compounds of formula I | 05-19-2011 |
20110166123 | NOVEL COMPOSITIONS AND METHODS OF USE - Described herein are novel enzyme inhibitors. In some embodiments the enzyme inhibitors are integrase inhibitors, particularly HIV integrase inhibitors. Also described herein are compositions containing them and methods of using them. Thus, the compounds and compositions described herein are useful for the in vitro and in vivo inhibition of HIV integrase as a method of treating or preventing HIV, AIDS or related disorders. | 07-07-2011 |
20110207812 | SUBSTITUTED ARYLAMINO-1,2,3,4-TETRAHYDRO NAPHTHALENES AND -2,3-DIHYDRO-1H-INDENES AS POTASSIUM CHANNEL MODULATORS - This invention provides compounds of formula I | 08-25-2011 |
20110269741 | NOVEL COMPOSITIONS AND METHODS OF USE - Described herein are novel enzyme inhibitors. In some embodiments the enzyme inhibitors are integrase inhibitors, particularly HIV integrase inhibitors. Also described herein are compositions containing them and methods of using them. Thus, the compounds and compositions described herein are useful for the in vitro and in vivo inhibition of HIV integrase as a method of treating or preventing HIV, AIDS or related disorders. | 11-03-2011 |
20120329869 | BENZYLOXY ANILIDE DERIVATIVES USEFUL AS POTASSIUM CHANNEL MODULATORS - The present invention relates to benzyloxyanilide derivatives having the following structural formula: | 12-27-2012 |
20140155389 | BICYCLIC INHIBITORS OF ALK - The present invention relates to compounds of formula (1) or pharmaceutical acceptable salts, wherein R | 06-05-2014 |
20140171429 | BICYCLIC INHIBITORS OF ALK - The present invention relates to compounds of formula (1) or pharmaceutical acceptable salts, Formula (1) wherein R | 06-19-2014 |
20140194418 | BICYCLIC CARBOXAMIDE INHIBITORS OF KINASES - Compounds of formula (I) or pharmaceutical acceptable salts are provided, wherein X | 07-10-2014 |