| Patent application number | Description | Published |
|---|
| 20080221166 | AMINOAMIDES AS OREXIN ANTAGONISTS - The present invention relates to compounds of formula I | 09-11-2008 |
| 20080249125 | HETEROCYCLIC DERIVATIVES AS OREXIN ANTAGONISTS - The present invention relates to compounds of formula | 10-09-2008 |
| 20080249180 | MALONAMIDES AS OREXIN ANTAGONISTS - The present invention relates to compounds of formula I | 10-09-2008 |
| 20080275021 | PYRROLIDINE DERIVATIVES AS DUAL NK1/NK3 RECEPTOR ANTAGONISTS - The invention relates to pyrrolidine derivatives of formula | 11-06-2008 |
| 20080306086 | PROLINAMIDE DERIVATIVES AS NK3 ANTAGONISTS - The present invention relates to a compound of formula I | 12-11-2008 |
| 20080306089 | PROLINAMIDE-TETRAZOLE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS - The present invention relates to a compound of formula I | 12-11-2008 |
| 20080312216 | PIPERAZINE AND [1,4]DIAZEPAN DERIVATIVES AS NK ANTAGONISTS - The present invention relates to a compound of formula I | 12-18-2008 |
| 20090005370 | ISOXAZOLE-IMIDAZOLE DERIVATIVES - The present invention is concerned isoxazole-imidazole derivatives having affinity and selectivity for GABA A α5 receptor binding site, their manufacture, pharmaceutical compositions containing them and their use for enhancing cognition or for the treatment of cognitive disorders like Alzheimer's disease. In particular, the present invention is concerned with aryl-isoxazol-4-yl-imidazole derivatives of formula I | 01-01-2009 |
| 20090036422 | MONOAMIDE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS - The present invention relates to compounds of formula | 02-05-2009 |
| 20090042896 | PYRROLIDINE ARYL-ETHER AS NK3 RECEPTOR ANTAGONISTS - The invention relates to a compound of formula I | 02-12-2009 |
| 20090054644 | PYRROLIDINE ARYL-ETHER AS NK3 RECEPTOR ANTAGONISTS - The invention relates to a compound of general formula | 02-26-2009 |
| 20090076081 | PIPERIDINE DERIVATIVES AS NK3 ANTAGONISTS - The invention relates to a compound of formula | 03-19-2009 |
| 20090143371 | ISOXAZOLE-PYRIDINE DERIVATIVES - The present invention is concerned with isoxazole-pyridine derivatives of formula I | 06-04-2009 |
| 20090143385 | ISOXAZOLO-PYRIDAZINE DERIVATIVES - The invention relates to isoxazolo-pyridazine compounds, in particular those of formula I as described above and to a pharmaceutically acceptable salts thereof, having affinity and selectivity for the GABA A α5 receptor binding site, their manufacture, pharmaceutical compositions containing them and their use as cognitive enhancers or for the treatment of cognitive disorders like Alzheimer's disease. | 06-04-2009 |
| 20090143407 | ISOXAZOLO-PYRAZINE DERIVATIVES - The invention relates to isoxazolo-pyrazine derivatives and their pharmaceutically acceptable salts having affinity and selectivity for the GABA A α5 receptor binding site, their manufacture, and pharmaceutical compositions containing them. The compounds of present invention are inverse agonists of GABA A α5. The invention also relates to methods for enhancing cognition and for treating cognitive disorders like Alzheimer's disease. | 06-04-2009 |
| 20090163485 | HETEROARYL DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS - The present invention relates to compounds of formula | 06-25-2009 |
| 20090197875 | ARYL-ISOXAZOLO-4-YL-OXADIAZOLE DERIVATIVES - The present invention is concerned with isoxazol-4-yl-oxadiazole derivatives of formula | 08-06-2009 |
| 20090203736 | PIPERIDINE SULPHONAMIDE DERIVATIVES - The present invention relates to piperidine sulphonamide derivatives of formula | 08-13-2009 |
| 20090306043 | PYRROLIDINE ETHER DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS - The present invention relates to compounds of formula I | 12-10-2009 |
| 20090312314 | HETEROAROMATIC MONOAMIDES AS OREXININ RECEPTOR ANTAGONISTS - The present invention is concerned with novel sulfonamides of formula | 12-17-2009 |
| 20090312327 | PYRROLIDINE DERIVATIVES AS NK2 RECEPTOR ANTAGONISTS - The present invention relates to compounds of formula I | 12-17-2009 |
| 20100029664 | PYRROLIDIN-3-YLMETHYL-AMINE AS OREXIN ANTAGONISTS - The present invention is concerned with novel sulfonamides of formula I | 02-04-2010 |
| 20100041886 | ISOXAZOLO-PYRAZINE DERIVATIVES - The invention relates to isoxazolo-pyrazine derivatives and their pharmaceutically acceptable salts having affinity and selectivity for the GABA A α5 receptor binding site, their manufacture, and pharmaceutical compositions containing them. The compounds of present invention are inverse agonists of GABA A α5. The invention also relates to methods for enhancing cognition and for treating cognitive disorders like Alzheimer's disease. | 02-18-2010 |
| 20100075954 | SUBSTITUTED IMIDAZO[1,5-A][1,2,4]TRIAZOLO[1,5-D][1,4]BENZODIAZEPINE DERIVATIVES - The present invention is concerned with a method of treating Alzheimer's disease by administering a therapeutically effective amount of a substituted imidazo[1,5-a][1,2,4]triazolo[1,5-d][1,4]benzodiazepine of formula I | 03-25-2010 |
| 20100113424 | N-BENZYL PYRROLIDINE DERIVATIVES - The present invention relates to a compound of formula I | 05-06-2010 |
| 20100125078 | QUINAZOLINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS - The present invention relates to a compounds of formula I | 05-20-2010 |
| 20100168088 | PYRROLIDINE DERIVATIVES AS NK-3 RECEPTOR ANTAGONISTS - The present invention relates to a compound of formula I | 07-01-2010 |
| 20100197697 | PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS - The present invention relates to a compounds of formula I | 08-05-2010 |
| 20100210659 | PYRROLIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS - The present invention relates to a compounds of formula I | 08-19-2010 |
| 20100286117 | PYRIDINES - The present invention is concerned with novel isoxazoles of formula I | 11-11-2010 |
| 20110021565 | PIPERIDINE DERIVATIVES AS NK3 ANTAGONISTS - The invention relates to a compound of formula | 01-27-2011 |
| 20110053948 | PYRROLIDINES AS NK3 RECEPTOR ANTAGONISTS - The present invention relates to a compounds of formula I | 03-03-2011 |
| 20110071154 | PYRROLIDIN-3-YLMETHYL-AMINE AS OREXIN ANTAGONISTS - The present invention is concerned with novel sulfonamides of formula I | 03-24-2011 |
| 20110144081 | PYRROLIDINE DERIVATIVES - The present invention relates to compounds of formula | 06-16-2011 |
| 20110152233 | PYRROLIDINE COMPOUNDS - The present application relates to compounds of formula | 06-23-2011 |
