Patent application number | Description | Published |
20090099228 | PYRAZOLO-TETRAHYDRO PYRIDINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS - The invention relates to novel pyrazolo-tetrahydropyridines compounds and their use as orexin receptor antagonists. | 04-16-2009 |
20090275588 | NOVEL SULFONAMIDE COMPOUNDS - The invention relates to novel sulfonamide compounds and their use as orexin receptor antagonists. | 11-05-2009 |
20100016401 | 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES - The invention relates to 3-aza-bicyclo[3.1.0]hexane derivatives of formula (I) wherein A, B, n, X, and R | 01-21-2010 |
20100029617 | 1,4,5,6,7,8-HEXAHYDRO-1,2,5-TRIAZA-AZULENE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS - The invention relates to 1,4,5,6,7,8-hexahydro-1,2,5-triaza-azulene derivatives and their use as orexin receptor antagonists. | 02-04-2010 |
20100069418 | 3-HETEROARYL (AMINO OR AMIDO)-1-(BIPHENYL OR PHENYLTHIAZOLYL) CARBONYLPIPERIDINE DERIVATIVES AS OREXIN RECEPTOR INHIBITORS - The invention relates to piperidine compounds of formula (I) wherein X-R | 03-18-2010 |
20100093740 | 5,6,7,8-TETRAHYDRO-IMIDAZO[1,5-A]PYRAZINE DERIVATIVES - The invention relates to 5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine derivatives of formula (I), wherein X represents CH | 04-15-2010 |
20100113531 | THIAZOLIDINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS - The invention relates to novel thiazolidine derivatives of the formula (I) wherein A and R | 05-06-2010 |
20100184808 | 3-AZA-BICYCLO[3.3.0]OCTANE COMPOUNDS - The invention relates to 3-aza-bicyclo[3.3.0]octane derivatives of the formula (I) wherein R | 07-22-2010 |
20100197733 | PYRROLIDINES AND PIPERIDINES AS OREXIN RECEPTOR ANTAGONISTS - The invention relates to compounds of formula (I) wherein Y, A, N and R | 08-05-2010 |
20100204285 | TRANS-3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES - The invention relates to novel trans-3-aza-bicyclo[3.1.0]hexane derivatives of formula (I), wherein A, B, n and R | 08-12-2010 |
20100222328 | 2-CYCLOPROPYL-THIAZOLE DERIVATIVES - The invention relates to selected 2-cyclopropyl-thiazole derivatives of the formula (I) wherein B, Y and R1 are as described in the description; to salts and especially pharmaceutically acceptable salts thereof, and to the use of such compounds use as medicaments, especially as orexin receptor antagonists. | 09-02-2010 |
20100222600 | AZETIDINE COMPOUNDS AS OREXIN RECEPTOR ANTAGONISTS - The invention relates to novel azetidine compounds of formula (I), wherein R | 09-02-2010 |
20110009401 | 2-AZA-BICYCLO[2.2.1]HEPTANE DERIVATIVES - The invention relates to novel 2-aza-bicyclo[2.2.1]heptane derivatives of formula (I), | 01-13-2011 |
20110009461 | 2-AZA-BICYCLO[3.3.0]OCTANE DERIVATIVES - The invention relates to 2-aza-bicyclo[3.3.0]octane derivatives of Formula (I) wherein A, B, and R | 01-13-2011 |
20110039857 | PIPERIDINE AND PYROOLIDINE COMPOUNDS - The invention relates to piperidine and pyrrolidine compounds of formula (I) | 02-17-2011 |
20110086889 | TETRAZOLE COMPOUNDS AS OREXIN RECEPTOR ANTAGONISTS - The invention relates to tetrazole compounds of formula (I) wherein X, Y, Z, R | 04-14-2011 |
20110105491 | THIAZOLIDINE COMPOUNDS AS OREXIN RECEPTOR ANTAGONISTS - The invention relates to thiazolidine derivatives of the formula (I) wherein A, B, and R | 05-05-2011 |
20110105514 | 5,6,7,8-TETRAHYDRO-IMIDAZO[1,5-A]PYRAZINE COMPOUNDS - The invention relates to 5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine derivatives of formula (I) wherein R | 05-05-2011 |
20110124636 | 2-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS - The invention relates to novel 2-aza-bicyclo[3.1.0]hexane derivatives of Formula (I) wherein A, B, n and R | 05-26-2011 |
20110263662 | 1,2-DIAMIDO-ETHYLENE DERIVATIVES AS OREXIN ANTAGONISTS - The invention relates to 1,2-diamido-ethylene derivatives of the formula (I) wherein R | 10-27-2011 |
20110281869 | TETRAHYDROISOQUINOLINES AS ANTIMALARIAL AGENTS - The invention relates to novel tetrahydroisoquinoline derivatives and their use as active ingredients in the preparation of pharmaceutical compositions. The invention also concerns related aspects including pharmaceutical compositions containing one or more of those compounds and their use as medicaments for the treatment or prevention of protozoal infections, such as especially malaria. | 11-17-2011 |
20120088759 | THIAZOLIDIN-4-ONE AND [1,3]-THIAZINAN-4-ONE COMPOUNDS AS OREXIN RECEPTOR ANTAGONISTS - The present invention relates to thiazolidin-4-one and [1,3]-thiazinan-4-one compounds of formula (I) wherein X, Y, R | 04-12-2012 |
20120101111 | NOVEL OXAZOLIDINONE DERIVIATIVES - The present invention relates to oxazolidinone derivatives of formula (I) wherein Y, R | 04-26-2012 |
20130065902 | 3-(HETEROARYL-AMINO)-1,2,3,4-TETRAHYDRO-9H-CARBAZOLE DERIVATIVES AND THEIR USE AS PROSTAGLANDIN D2 RECEPTOR MODULATORS - The present invention relates to 3-(heteroaryl-amino)-1,2,3,4-tetrahydro-9H-carbazole derivatives of the formula (I), | 03-14-2013 |
20130237525 | LACTAM DERIVATIVES USEFUL AS OREXIN RECEPTOR ANTAGONISTS - The present invention relates to lactam derivatives of formula (I) | 09-12-2013 |