Patent application number | Description | Published |
20080207647 | Pyrazole Derivatives Having Tyrosine Kinase Activity - Compounds of the formula (I), in which R, X, R | 08-28-2008 |
20080207682 | Phenylurea Derivatives As Inhibitors Of Tyrosine Kinases For The Treatment Of Tumour Diseases - Compounds of the formula (I), in which R | 08-28-2008 |
20080207699 | Pyrazole Derivatives -
Compounds of the formula (I), in which R | 08-28-2008 |
20080214582 | Purine Derivatives as Inhibitors of Receptor Tyrosine Kinase Activity - Compounds of the formula (I), in which R | 09-04-2008 |
20080306042 | Triazole Derivatives - Novel triazole derivatives are inhibitors of TGF-beta receptor I kinase, and can be employed, inter alia, for the treatment of tumours. | 12-11-2008 |
20090215799 | HETEROCYCLIC SUBSTITUTED BISARYLUREA DERIVATIVES - The present invention relates to heterocyclic substituted bisarylurea derivatives of formula I, the use of the compounds of formula I as inhibitors of one or more kinases, the use of the compounds of formula I for the manufacture of a pharmaceutical composition and a method of treatment, comprising administering said pharmaceutical composition to a patient. | 08-27-2009 |
20100063028 | Triazabenzo[E]Azulene Derivatives for the Treatment Of Tumors - Novel triazabenzo[e]azulene derivatives of the formula, (I) in which R | 03-11-2010 |
20100234369 | 5-CYANOTHIENOPYRIDINES FOR THE TREATMENT OF TUMOURS - Novel 5-cyanothienopyridines of the formula (I), in which R | 09-16-2010 |
20110028472 | THIENOPYRIMIDINES - Novel thienopyrimidines of the formula (I), in which R | 02-03-2011 |
20110130396 | IMIDAZOTHIADIAZOLE DERIVATIVES - Novel imidazo[2,1-b][1,3,4]thiadiazole derivatives of formula (I) | 06-02-2011 |
20120101095 | ALKOXY-THIENOPYRIMIDINES AS TGF-BETA RECEPTOR KINASE MODULATORS - Novel alkoxy-thienopyrimidine derivatives of formula (I) | 04-26-2012 |
20120295902 | Hetaryl-[1,8]naphthyridine derivatives - Novel hetaryl-[1,8]naphthyridine derivatives of formula (I) | 11-22-2012 |
20130102603 | 2,4-DIARYL - SUBSTITUTED [1,8] NAPHTHYRIDINES AS KINASE INHIBITORS FOR USE AGAINST CANCER - The present invention relates to novel [1,8]naphthyridine derivatives of formula (I) and to the use of such compounds in which the inhibition, regulation and/or modulation of signal transduction by ATP consuming proteins like kinases plays a role, particularly to inhibitors of TGF-beta receptor kinases, and to the use of such compounds for the treatment of kinase-induced diseases, in particular for the treatment of tumors. | 04-25-2013 |
20130102608 | BIPYRIDYL DERIVATIVES - The present invention relates to novel bipyridyl derivatives of formula (I) and to the use of such compounds in which the inhibition, regulation and/or modulation of signal transduction by ATP consuming proteins like kinases plays a role, particularly to inhibitors of TGF-beta receptor kinases, and to the use of such compounds for the treatment of kinase-induced diseases, in particular for the treatment of tumors. | 04-25-2013 |
20130345227 | PYRIDO [2, 3 - B] PYRAZINE DERIVATIVES AND THEIR THERAPEUTICAL USES - The present invention relates to novel pyrido[2,3-b]pyrazine derivatives of formula (I) and to the use of such compounds in which the inhibition, regulation and/or modulation of signal transduction by ATP consuming proteins like kinases plays a role, particularly to inhibitors of TGF-beta receptor kinases, and to the use of such compounds for the treatment of kinase-induced diseases, in particular for the treatment of tumors. | 12-26-2013 |
20140038960 | Hetaryl-[1,8]naphthyridine derivatives - Novel hetaryl-[1,8]naphthyridine derivatives of formula (I) | 02-06-2014 |
20140142097 | PYRIDINE-AND PYRAZINE DERIVATIVES - Compounds of the formula (I) in which R, R | 05-22-2014 |
20140323481 | 3-CYANOARYL-1H-PYRROLO[2,3-B]PYRIDINE DERIVATIVES - Compounds of the formula (I) in which R | 10-30-2014 |
20140336201 | BIPYRIDYL DERIVATIVES - The present invention relates to novel bipyridyl derivatives of formula (I) and to the use of such compounds in which the inhibition, regulation and/or modulation of signal transduction by ATP consuming proteins like kinases plays a role, particularly to inhibitors of TGF-beta receptor kinases, and to the use of such compounds for the treatment of kinase-induced diseases, in particular for the treatment of tumors. | 11-13-2014 |
20140378431 | TRIAZOLO[4,5-D]PYRIMIDINE DERIVATIVES - Compounds of the formula I | 12-25-2014 |
20150051202 | TRIAZOLOPYRAZINE DERIVATIVES - Compounds of the formula I | 02-19-2015 |