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Gregor James Macdonald
Gregor James Macdonald, Harlow GB
| Patent application number | Description | Published |
|---|---|---|
| 20080214571 | NOVEL COMPOUNDS - Disclosed is a method for use of phenyl sulfone compounds of formula (I) in the treatment of anxiety. | 09-04-2008 |
| 20090012099 | Novel Compounds - Disclosed is a method for use of phenyl sulfone compounds of formula (I) in the treatment of Alzheimer's disease and age related cognitive decline. | 01-08-2009 |
| 20090036682 | Quinoline Derivatives and Their Use as 5-HT6 Ligands - The present invention relates to novel quinoline compounds having pharmacological activity, to processes for their preparation, to compositions containing them and to their use in the treatment of CNS and other disorders. | 02-05-2009 |
| 20100305107 | QUINOLINE DERIVATIVES AND THEIR USE AS 5-HT6 LIGANDS - Disclosed are quinoline compounds having affinity for the 5-HT | 12-02-2010 |
| 20110237792 | QUINOLINE DERIVATIVES AND THEIR USE AS 5-HT6 LIGANDS - Disclosed are quinoline compounds having affinity for the 5-HT | 09-29-2011 |
Gregor James Macdonald, Beerse BE
| Patent application number | Description | Published |
|---|---|---|
| 20100166655 | 1, 4-DISUBSTITUTED 3-CYANO-PYRIDONE DERIVATIVES AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF MGLUR2-RECEPTORS - The present invention relates to novel compounds, in particular novel pyridinone derivatives according to Formula (I) | 07-01-2010 |
| 20100240688 | 1,3-DISUBSTITUTED-4-PHENYL-3,4,5,6-TETRAHYDRO-2H,1 H-1,4 BIPYRIDINYL-2-ONES - The present invention relates to novel compounds, in particular novel pyridinone derivatives according to Formula (I) | 09-23-2010 |
| 20100240706 | 1,3-DISUBSTITUTED-4-PHENYL-1H-PYRIDIN-2-ONES - The present invention relates to novel compounds, in particular novel pyridinone derivatives according to Formula (I) | 09-23-2010 |
| 20100286206 | 1,3-DISUBSTITUTED 4-(ARYL-X-PHENYL)-1H-PYRIDIN-2-ONES - The present invention relates to novel compounds, in particular novel pyridinone derivatives according to Formula (I) | 11-11-2010 |
Gregor James Macdonald, Zoersel GB
| Patent application number | Description | Published |
|---|---|---|
| 20100063092 | 3-CYANO-4-(4-PHENYL-PIPERIDIN-1-YL)-PYRIDIN-2-ONE DERIVATIVES - The present invention relates to novel compounds, in particular novel pyridinone derivatives according to Formula (I) including any stereochemically isomeric form thereof, or a pharmaceutically acceptable salt thereof or a solvate thereof, wherein all radicals are defined in the application and claims. The compounds according to the invention are positive allosteric modulators of metabotropic glutamate receptors subtype 2 (“mGluR2”) which are useful for the treatment or prevention of neurological and psychiatric disorders associated with glutamate dysfunction and diseases in which the mGluR2 subtype of metabotropic receptors is involved. In particular, such diseases are central nervous system disorders selected from the group of anxiety, schizophrenia, migraine, depression, and epilepsy. The invention is also directed to pharmaceutical compositions and processes to prepare such compounds and such compositions, as well as to the use of such compounds for the prevention and treatment of such diseases in which mGluR2 is involved. | 03-11-2010 |
Gregor James Macdonald, Essex GB
| Patent application number | Description | Published |
|---|---|---|
| 20080306083 | Biaryl Compounds Useful as Agonists of the Gpr38 Receptor - The present invention relates to novel biaryl derivatives such as compounds of formula (I), which have activity as agonists of the GPR38 receptor and the use of such compounds or pharmaceutical compositions thereof in the treatment of gastrointestinal disorders. | 12-11-2008 |
| 20080312209 | Piperazine Heteroaryl Derivatives as Gpr38 Agonists - The invention provides compounds of formula (I) or pharmaceutically acceptable salts thereof, | 12-18-2008 |
| 20090298841 | QUINOLINE DERIVATIVES AND THEIR USE AS 5-HT6 LIGANDS - The present invention relates to novel quinoline compounds having pharmacological activity, to processes for their preparation, to compositions containing them and to their use in the treatment of CNS and other disorders. | 12-03-2009 |
Gregor James Macdonald, Emblem BE
| Patent application number | Description | Published |
|---|---|---|
| 20080227791 | Piperidin-4-Yl-Pyridazin-3-Ylamine Derivatives as Fast Dissociating Dopamine 2 Receptor Antagonists - The present invention relates to compounds that are fast dissociating dopamine 2 receptor antagonists, processes for preparing these compounds, pharmaceutical compositions comprising these compounds as an active ingredient. The compounds find utility as medicines for treating or preventing central nervous system disorders, for example schizophrenia, by exerting an antipsychotic effect without motor side effects. | 09-18-2008 |
Gregor James Macdonald, Ranst BE
| Patent application number | Description | Published |
|---|---|---|
| 20110269748 | 2-ANILINE-4-ARYL SUBSTITUTED THIAZOLE DERIVATIVES - This invention concerns the use of a compound of formula (I) | 11-03-2011 |