Patent application number | Description | Published |
20080214598 | Novel Piperidine Carboxylic Acid Amide Derivatives - The invention relates to novel piperidine carboxylic acid amide derivatives and their use as active ingredients in the preparation of pharmaceutical compositions. The invention also concerns related aspects including processes for the preparation of these novel compounds, pharmaceutical compositions comprising such compounds and especially the use of such compounds as inhibitors of renin. | 09-04-2008 |
20090306123 | Bicyclononene derivaties - The invention relates to novel bicyclononene derivatives of Formula (I); and the use thereof as active ingredients in the preparation of pharmaceutical compositions. The invention also concerns related aspects including processes for the preparation of the compounds, pharmaceutical compositions containing one or more of those compounds and especially their use as inhibitors of renin. | 12-10-2009 |
20120101138 | FLUORINATED AMINOTRIAZOLE DERIVATIVES - The invention relates to fluorinated aminotriazole derivatives of formula (I), | 04-26-2012 |
20120115841 | BRIDGED SPIRO [2.4] HEPTANE DERIVATIVES AS ALX RECEPTOR AND/OR FPRL2 AGONISTS - The present invention relates to bridged spiro[2.4]heptane derivatives of formula (I), wherein W, Y, Z, R | 05-10-2012 |
20120115916 | OXAZOLE AND THIAZOLE DERIVATIVES AS ALX RECEPTOR AGONISTS - The invention relates to oxazole and thiazole derivatives of formula (I), wherein A, E, X, R | 05-10-2012 |
20130096119 | Isoquinolin-3-Ylurea Derivatives - The invention relates to isoquinolin-3-ylurea derivatives of formula (I) wherein R | 04-18-2013 |
20130231319 | Bridged Spiro[2.4]heptane Ester Derivatives - The invention relates to a method for preparing linear polymers having an amide end or having a star architecture comprising an amide core, by means of a ring opening using lactide and glycolide monomers or a lactide monomer ring in the presence of a catalyst, wherein the method includes the steps of: (i) reacting the excess monomer(s) with an initiator in a solvent, said initiator being selected from among an amine and an amino alcohol, given that the initiator has at least one primary or secondary amine function; (ii) adding a catalyst, said catalyst being a non-nucleophilic base and including at least one neutral sp2 nitrogen atom; and (iii) neutralizing the reaction mixture. Said novel method is particularly advantageous in that it can be easily monitored and enables better modulation of the polymers, and thus of the properties thereof, than the methods of the prior art. The invention also relates to novel polymers that are obtainable by means of said method. | 09-05-2013 |
20130261159 | OXAZOLYL-METHYLETHER DERIVATIVES AS ALX RECEPTOR AGONISTS - The invention relates to oxazolyl-methylether derivatives of formula (I), | 10-03-2013 |
20130267569 | Hydroxylated Aminotriazole Derivatives as ALX Receptor Agonists - The invention relates to hydroxylated aminotriazole derivatives of formula (I), | 10-10-2013 |