Buijnsters
Peter Jacobus Johannes Buijnsters, Etten-Leur NL
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20110009404 | 4-ARYL-2-ANILINO-PYRIMIDINES - The present invention relates to compounds of Formula (Ia) or (Ib), the N-oxide forms, pharmaceutically acceptable addition salts, quaternary amines, stereoisomers, tautomers, racemics, metabolites, prodrugs, hydrates, or solvates thereof, | 01-13-2011 |
Peter Jacobus Johannes Buijnsters, Beerse BE
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20130197022 | 3-CYANO-QUINOLINE DERIVATIVES WITH ANTIPROLIFERATIVE ACTIVITY - The present invention concerns the compounds of formula | 08-01-2013 |
Peter Jacobus Johannes Buijnsters, Breda BE
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20140256948 | 3-CYANO-QUINOLINE DERIVATIVES WITH ANTIPROLIFERATIVE ACTIVITY - The present invention concerns the compounds of formula | 09-11-2014 |
Peter Jacobus Johannes Antonius Buijnsters, Etten Leur BE
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20100190786 | INDOLIN-2-ONES AND AZA-INDOLIN-2-ONES - The present invention relates to compounds or pharmaceutically-acceptable salts thereof, processes for preparing them, pharmaceutical compositions containing them and their use in therapy. The invention particularly relates to certain indolin-2-ones and aza-indolin-2-ones which possess anti-tumour activity and are accordingly useful in methods of treatment of the human or animal body, in particular such compounds are useful in the treatment of pathological processes which involve an aberrant cellular proliferation, such as tumor growth, rheumatoid arthritis, restenosis and atherosclerosis. | 07-29-2010 |
Peter Jacobus Johannes Antonius Buijnsters, Breda NL
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20090036471 | Triazolopyrimidine Derivatives As Glycogen Synthase Kinase 3 Inhibitors - This invention concerns compounds of formula | 02-05-2009 |
20100069424 | 3-CYANO-QUINOLINE DERIVATIVES WITH ANTIPROLIFERATIVE ACTIVITY - The present invention concerns the compounds of formula | 03-18-2010 |
20100105668 | Quinazoline derivatives - The present invention concerns the compounds of formula | 04-29-2010 |
20100173913 | PYRIDO-AND PYRIMIDOPYRIMIDINE DERIVATIVES AS ANTI-PROLIFERATIVE AGENTS - The present invention concerns the compounds of formula | 07-08-2010 |
20130178624 | QUINAZOLINE DERIVATIVES - The present invention concerns the compounds of formula | 07-11-2013 |
Peter Jacobus Johannes Antonius Buijnsters, Beerse BE
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20140147386 | 1-ARYL-4-METHYL-[1,2,4]TRIAZOLO[4,3-a]QUINOXALINE DERIVATIVES - The present invention relates to novel 1-aryl-4-methyl-[1,2,4]triazolo[4,3-a]-quinoxaline derivatives as inhibitors of phosphodiesterase 2 (PDE2) and to a lesser extent of phosphodiesterase 10 (PDE10) or as inhibitors of both, phosphodiesterases 2 and 10. The invention is also directed to pharmaceutical compositions comprising such compounds, to processes for preparing such compounds and compositions, and to the use of such compounds and compositions for the prevention and treatment of disorders in which PDE2 is involved, or disorders in which both PDE2 and PDE 10 are involved, such as neurological and psychiatric disorders, and endocrinological or metabolic diseases. The present invention also relates to radiolabelled compounds which may be useful for imaging and quantifying the PDE2 enzyme in tissues, using positron-emission tomography (PET). The invention is also directed to compositions comprising such compounds, to processes for preparing such compounds and compositions, to the use of such compounds and compositions for imaging a tissue, cells or a host, in vitro or in vivo and to precursors of said compounds. | 05-29-2014 |