Patent application number | Description | Published |
20080300290 | Novel Beta-Agonists, Process for Their Preparation and Their Use as Medicaments - Compounds of general formula (I) | 12-04-2008 |
20090111797 | Selected CGRP-antagonists, process for preparing them and their use as pharmaceutical compositions - The present invention relates to the CGRP antagonists of general formula | 04-30-2009 |
20090176770 | Selected CGRP-antagonists, process for preparing them and their use as pharmaceutical compositions - The present invention relates to the CGRP antagonists of general formula | 07-09-2009 |
20090186881 | CGRP-antagonists, process for preparing them and their use as pharmaceutical compositions - The present invention relates to the CGRP-antagonists of general formula I | 07-23-2009 |
20090253680 | SELECTED CGRP-ANTAGONISTS, PROCESSES FOR PREPARING THEM AND THEIR USE AS PHARMACEUTICAL COMPOSITIONS - The present invention relates to the CGRP-antagonists of general formula I | 10-08-2009 |
20100004228 | SELECTED CGRP ANTAGONISTS, PROCESSES FOR PREPARING THEM AND THEIR USE AS PHARMACEUTICAL COMPOSITIONS - The present invention relates to the CGRP antagonists of general formula I | 01-07-2010 |
20100144716 | New CGRP-antagonists, process for preparing them and their use as pharmaceutical compositions - The present invention relates to the CGRP-antagonists of general formula I | 06-10-2010 |
20100222336 | SINGLE ENANTIOMER BETA-AGONISTS, METHODS FOR THE PRODUCTION THEREOF AND THE USE THEREOF AS MEDICATION - The present invention relates to single enantiomer compounds of formula (1), where the moieties n, A, R | 09-02-2010 |
20100234361 | SELECTED CGRP-ANTAGONISTS, PROCESS FOR PREPARING THEM AND THEIR USE AS PHARMACEUTICAL COMPOSITIONS - The present invention relates to the CGRP antagonists of general formula | 09-16-2010 |
20100249114 | Selected CGRP-antagonists, process for preparing them and their use as pharmaceutical compositions - The present invention relates to the CGRP antagonists of general formula | 09-30-2010 |
20110034444 | SELECTED CGRP ANTAGONISTS, PROCESSES FOR PREPARING THEM AND THEIR USE AS PHARMACEUTICAL COMPOSITIONS - The present invention relates to the CGRP antagonists of general formula I | 02-10-2011 |
20110183987 | Stereoselective Synthesis of Bicyclic Heterocycles - The present invention relates to a process for the stereoselective preparation of compounds of formulae (1A) and (1B) | 07-28-2011 |
20110262369 | CRYSTALLINE, ENANTIOMERICALLY PURE SALT FORM OF A BETA-AGONIST, AND THE USE THEREOF AS A DRUG - The invention relates to a crystalline, enantiomerically pure hydrochloride salt of N-(5-{2-[3-(4,4-diethyl-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-1,1-dimethyl-propylamino]-1-hydroxy-ethyl}-2-hydroxy-phenyl)-methane sulfonamide, preferably N-(5-{(R)-2-[3-(4,4-diethyl-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-1,1-dimethyl-propylamino]-1-hydroxy-ethyl}-2-hydroxy-phenyl)-methane sulfonamide, and the effect thereof as a long-term betamimetic agent, alone or combined with at least one other active ingredient, in the treatment of respiratory diseases. | 10-27-2011 |
20120004252 | NEW CCR2 RECEPTOR ANTAGONISTS AND USES THEREOF - The present invention relates to novel antagonists for CCR2 (CC chemokine receptor 2) and their use for providing medicaments for treating conditions and diseases, especially pulmonary diseases like asthma and COPD. | 01-05-2012 |
20120046284 | Salts and hydrates of 4-[(3-chloro-4-fluoro-phenyl)amino]-6-(cis-4--cyclohexan-1-yloxy)-7-metho- xy-quinazoline, their use as a medicament and the preparation thereof - The present invention relates to a compound of formula (I), | 02-23-2012 |
20120264729 | CO-CRYSTALS AND SALTS OF CCR3-INHIBITORS - This invention relates to co-crystals and salts of CCR3 inhibitors of formula 1, | 10-18-2012 |
20130143905 | NOVEL ANTAGONISTS FOR CCR2 AND USES THEREOF - The present invention relates to novel antagonists for CCR2 (CC chemokine receptor 2) of formula (I) and their use for providing medicaments for treating conditions and diseases, especially pulmonary diseases like asthma and COPD. | 06-06-2013 |
20140135307 | CO-CRYSTALS AND SALTS OF CCR3-INHIBITORS - This invention relates to co-crystals and salts of CCR3 inhibitors of formula 1, | 05-15-2014 |
20140135495 | STEREOSELECTIVE SYNTHESIS OF BICYCLIC HETEROCYCLES - The present invention relates to a process for the stereoselective preparation of compounds of formulae (1A) and (1B) | 05-15-2014 |
20140235661 | NEW CCR2 RECEPTOR ANTAGONISTS AND USES THEREOF - The present invention relates to novel antagonists for CCR2 (CC chemokine receptor 2) and their use for providing medicaments for treating conditions and diseases, especially pulmonary diseases like asthma and COPD. | 08-21-2014 |
20150087829 | PROCESS AND INTERMEDIATES FOR PREPARING GPR40 AGONISTS - The present invention relates to compounds of formula I | 03-26-2015 |