Patent application number | Description | Published |
20100029987 | Crystalline Form of Rasagiline and Process for the Preparation Thereof - A process for the preparation of (R)—N-propargyl-1-aminoindane, or a salt thereof, comprising reacting 1-indanone with propargylamine, in presence of a mixture of sodium borohydride and acetic acid, to obtain N-propargyl-1-aminoindane; and its conversion into (R)—N-propargyl-1-aminoindane or a salt thereof. | 02-04-2010 |
20100228034 | PROCESS FOR THE PREPARATION OF KETO INTERMEDIATES - Process for the preparation of 4-[1-oxo-4-[4-(hydroxyphenylmethyl)-1-piperidinyl]butyl]-α,α-dimethylbenzenacetic acid, which is an intermediate useful in the preparation of fexofenadine, by hydrating asymmetric alkynes. | 09-09-2010 |
20100234616 | METHOD FOR THE PREPARATION OF RUFINAMIDE - The invention provides a novel process for the regioselective preparation of a compound of formula (I) | 09-16-2010 |
20100267954 | PROCESS FOR THE PURIFICATION OF PALIPERIDONE - Process for the purification of paliperidone by formation of a salt thereof, such as the hydrochloride. | 10-21-2010 |
20100292506 | PROCESS FOR THE SYNTHESIS OF PREGABALIN - A process for the preparation of a compound of formula (I) is disclosed, | 11-18-2010 |
20100297711 | PROCESS FOR THE SYNTHESIS OF FOSINOPRIL AND INTERMEDIATES THEREOF - Process for the preparation of intermediates useful in the synthesis of [1[S(R)],2α,4β]-4-cyclohexyl-1-[[[(2-methyl-1-oxypropoxy)propoxy](4-phenylbutyl)phosphinyl]acetyl]-L-proline, and the synthesis thereof, in particular as sodium salt. | 11-25-2010 |
20100331541 | PROCESS FOR THE PREPARATION OF SITAGLIPTIN - A process for the preparation of 2(R)-4-oxo-4-[3-(trifluoromethyl)-5,6-dihydro[1,2,4]triazolo[4,3-a]-7(8H)-pyrazinyl]-1-(2,4,5-trifluorophenyl)-2-butanamine and intermediates useful for the synthesis thereof. | 12-30-2010 |
20120142939 | PROCESS FOR THE PREPARATION OF FOSINOPRIL AND INTERMEDIATES THEREOF - The present invention relates to a process for the preparation of intermediates useful in the synthesis of [1[S(R)],2α,4β]-4-cyclohexyl-1-[[[2-methyl-1-oxypropoxy)propoxy](4-phenylbutyl phosphinyl]acetyl]L-proline, and the synthesis thereof, in particular as sodium salt (fosinopril sodium). | 06-07-2012 |
20120149772 | PROCESS FOR THE PREPARATION OF FESOTERODINE OR A SALT THEREOF - A process for the preparation of (R)-2-(3-diisopropylamino-1-phenylpropyl)-4-(hydroxymethyl)-phenol isobutyrate (Fesoterodine) or a pharmaceutically acceptable salt thereof having low content in impurities. | 06-14-2012 |
20120165525 | PROCESS FOR THE PREPARATION OF LINAGLIPTIN - The present invention relates to processes for the preparation of 8-(3R)-3-aminopiperidinyl)-7-butyn-2-yl-3 -methyl-1-(4-methyl-quinazolin-2-ylmethyl)-3,7-dihydropurine-2,6-dione and novel intermediates useful in its synthesis. | 06-28-2012 |
20120277443 | PROCESS FOR THE PURIFICATION OF RUFINAMIDE - A process for purifying Rufinamide, comprising: | 11-01-2012 |
20130030179 | PROCESS FOR THE PREPARATION OF VARENICLINE - It is disclosed a process for the preparation of a compound of formula (I) or a salt thereof, comprising: | 01-31-2013 |
20140148574 | SYNTHESIS OF AN INTERMEDIATE OF AN ANTIVIRAL COMPOUND - Process for the preparation of a cyclopropylamide compound which is useful as a structural unit in a process for the preparation of a viral protease inhibitor. | 05-29-2014 |
20140275610 | PROCESS FOR THE PREPARATION OF FESOTERODINE OR A SALT THEREOF - A process for the preparation of (R)-2-(3-diisopropylamino-1-phenylpropyl)-4-(hydroxymethyl)-phenol isobutyrate (Fesoterodine) or a pharmaceutically acceptable salt thereof having low content in impurities. | 09-18-2014 |
Patent application number | Description | Published |
20130090474 | PROCESS FOR THE PREPARATION OF PTERIDINE DERIVATIVES - The application discloses a process for the preparation of 5-deoxy-L-arabinose of formula (VI); comprising the conversion of a compound of formula (XII); wherein n is 0, 1 or 2; which can be used as intermediate for the synthesis of sapropterin. | 04-11-2013 |
20140275542 | SYNTHESIS OF A SEROTONIN REUPTAKE INHIBITOR - Process for the preparation of a piperazinyl derivative, and its intermediates, which has known activity as a serotonin reuptake inhibitor and is used in therapy for treating serious symptoms of depression in adults. | 09-18-2014 |
20140303402 | PROCESS FOR THE PREPARATION OF SULFONAMIDE COMPOUNDS - Process for the preparation of known sulfonamides having antibacterial activity applicable on industrial scale, which allows their production in high yields and purity, comprising in particular the step of nucleophile aromatic substitution and oxidation in suitable conditions. | 10-09-2014 |
20150099899 | PROCESS FOR THE PURIFICATION OF 2-PHENYL-2-METHYL-PROPANOIC ACID DERIVATIVES - Process for the preparation of 2-phenyl-2-methyl propanoic acid derivatives, useful as intermediates in the preparation of fexofenadine hydrochloride. | 04-09-2015 |
20150111934 | CRYSTALLINE FORMS OF AN ADRENERGIC AGONIST - The present invention relates to the acetate salt of Mirabegron, in particular in two novel crystalline forms, a process for their preparation and the use of said salt and its crystalline forms in the synthesis of Mirabegron with high yields and chemical purity. | 04-23-2015 |