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DIPHARMA FRANCIS S.R.L.

DIPHARMA FRANCIS S.R.L. Patent applications
Patent application numberTitlePublished
20110269962PROCESS FOR PREPARING STATINS - Process for the preparation of β-ketoester synthetic intermediates useful in the preparation of statins, in particular Pitavastatin.11-03-2011
20110152367PROCESS FOR THE PREPARATION OF FESOTERODINE WITH LOW IMPURITIES CONTENT - Disclosed is a process for the preparation of (R)-2-(3-diisopropylamino-1-phenylpropyl)-4-(hydroxymethyl)-phenol isobutyrate (Fesoterodine) or a pharmaceutically acceptable salt thereof having a low content of impurities such as tolterodine and tolterodine isobutyrate.06-23-2011
20110124917PROCESS FOR THE PREPARATION OF CINACALCET AND INTERMEDIATES THEREOF - The present invention relates to a process for the preparation of (R)-(1-Naphthalen-1-yl-ethyl)-[3-(3-trifluoromethyl-phenyl)-propyl]-amine or a salt thereof, in particular the hydrochloride, and intermediates useful in its synthesis.05-26-2011
20110034523CRYSTALLINE FORMS OF RUFINAMIDE - Disclosed is a crystalline form of rufinamide selected from: 02-10-2011
20110028728PROCESS FOR THE PREPARATION OF CRYSTALLINE DEXLANSOPRAZOLE - Process for the preparation of crystalline anhydrous (R)-2-[[[3-methyl-4-(2,2,2-trifluoroetoxy)-2-piridyl]methyl]sulphinyl]benzimidazole (dexlansoprazole).02-03-2011
20100331541PROCESS FOR THE PREPARATION OF SITAGLIPTIN - A process for the preparation of 2(R)-4-oxo-4-[3-(trifluoromethyl)-5,6-dihydro[1,2,4]triazolo[4,3-a]-7(8H)-pyrazinyl]-1-(2,4,5-trifluorophenyl)-2-butanamine and intermediates useful for the synthesis thereof.12-30-2010
20100297711PROCESS FOR THE SYNTHESIS OF FOSINOPRIL AND INTERMEDIATES THEREOF - Process for the preparation of intermediates useful in the synthesis of [1[S(R)],2α,4β]-4-cyclohexyl-1-[[[(2-methyl-1-oxypropoxy)propoxy](4-phenylbutyl)phosphinyl]acetyl]-L-proline, and the synthesis thereof, in particular as sodium salt.11-25-2010
20100292506PROCESS FOR THE SYNTHESIS OF PREGABALIN - A process for the preparation of a compound of formula (I) is disclosed,11-18-2010
20100267954PROCESS FOR THE PURIFICATION OF PALIPERIDONE - Process for the purification of paliperidone by formation of a salt thereof, such as the hydrochloride.10-21-2010
20100234616METHOD FOR THE PREPARATION OF RUFINAMIDE - The invention provides a novel process for the regioselective preparation of a compound of formula (I)09-16-2010
20090312550ZIPRASIDONE FREE FROM COLORED IMPURITIES AND A PROCESS FOR ITS PREPARATION - Ziprasidone base or a pharmaceutically acceptable salt thereof free from colored impurities, in particular those giving the product a “slightly pink to pink” coloration.12-17-2009
20090203915Process for the preparation of solifenacin - A process for the preparation of (1S,3′R)-quiniclidin-3′-yl-1-phenyl-3,4-dihydro-1H-isoquinolin-2-carboxylate, namely solifenacin, comprising the reaction of a compound of formula (IV) with a compound of formula (V), as herein defined,08-13-2009
20090156855CRYSTALLINE FORM OF (S)-1-PHENYLETHYLAMMONIUM (R)-DIPHENYLMETHANESULPHINYL-ACETATE - Novel crystalline hydrate form of (S)-1-phenylethylammonium (R)-diphenyl-methanesulphinyl-acetate and its use in a process for the preparation of (R)-benzhydrylsulphinylacetamide.06-18-2009
20090156811Process for the Preparation of Bosentan - A process for the preparation of 4-tert-butyl-N-[6-(2-hydroxy-ethoxy)-5-(2-methoxy-phenoxy)-[2,2′]bipyrimidinyl-4-yl]-benzenesulfonamide, bosentan, comprising the reaction of a compound of formula (II) or a salt thereof,06-18-2009
20090143615Process for the Preparation of (S)(+)-3-(Aminomethyl)-5-Methylhexanoic Acid - A process for the preparation of a compound of formula (I),06-04-2009
20090076277Process for the preparation of pyridine-methylsulfinyl compounds - A process for the preparation of a compound of formula (I), or a salt thereof,03-19-2009
20090062534LINEZOLID CRYSTALLINE HYDRATE FORM AND LINEZOLID SALTS - Linezolid salts, useful as such and as intermediates in a process for the preparation of novel and known crystalline linezolid forms, in particular known as Form III.03-05-2009
20080319229 PROCESS FOR THE PREPARATION OF CINACALCET - The invention provides a novel process for the preparation of a compound of formula (I)12-25-2008
20080311635PROCESS FOR THE PREPARATION OF (S)(+)-3-(AMINOMETHYL)-5-METHYLHEXANOIC ACID - A process for the preparation of (S)(+)-3-(aminomethyl)-5-methylhexanoic acid (pregabalin) of formula (I) or a salt thereof,12-18-2008
20080293948PROCESS FOR THE PREPARATION OF KETO COMPOUNDS - A process for the preparation of 4-[1-oxo-4-[4-(hydroxydiphenylmethyl)-1-piperidinyl]butyl]-α,α-dimethylbenzeneacetic acid, useful as an intermediate for the preparation of fexofenadine, is provided.11-27-2008

Patent applications by DIPHARMA FRANCIS S.R.L.