| CarboDesign LLC Patent applications |
| Patent application number | Title | Published |
| 20110137047 | Process for enantiomerically pure 8-Aryloctanoic acids as Aliskiren - The present invention relates to a novel manufacturing process and novel intermediates useful in the synthesis of pharmaceutically active compounds, especially rennin inhibitors such as Aliskiren. The invention describes a preparation of enantiomerically pure 8-aryloctanoic acids of general formula I from readily available key intermediate, chiral cis-diacid of formula II, aziridine of formula XI and a monocyclic compound of formula III. | 06-09-2011 |
| 20110105767 | Manufacturing process for enantiomerically pure 8-Aryloctanoic acids as Aliskiren - The invention describes a novel technical process and novel intermediates useful for the manufacture of enantiomerically pure 8-aryloctanoic acids of the formula I which are pharmaceutically active compounds as rennin inhibitors. | 05-05-2011 |
| 20110092706 | Process for the manufacture of enantiomerically pure aryloctanoic acids as aliskiren - The present invention relates to a novel manufacturing process and novel intermediates useful in the synthesis of pharmaceutically active compounds, especially rennin inhibitors such as Aliskiren. The invention describes a preparation of enantiomerically pure 8-aryloctanoic acids of general formula I from readily available key intermediate, a novel bicyclic compound of formula IV. | 04-21-2011 |